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AT13148 1056901-62-2 AT13148 is a novel oral multi-AGC kinase inhibitor with potent pharmacodynamic and antitumor activity, which shows a distinct mechanism of action from other AKT inhibitors.
K-115 223645-67-8 K-115 (free base)是一高效选择性ROCK激酶抑制剂,IC50值为31nM。
GSK269962A(GSK269962) 850664-21-0 GSK269962A(GSK269962)是人ROCK1和ROCK2抑制剂,IC50分别为1.6和4 nM,比对其它丝an酸/苏an酸激酶的抑制性强30倍。
AR-13324 hydrochloride 1253952-02-1 AR-13324是ROCK抑制剂,Ki值为0.2-10.3 nM。
Fasudil hydrochloride 105628-07-7 Fasudil Hydrochloride (盐suan法舒地尔; HA-1077; AT-877) 能抑制ROCK-II,PKA,PKG,PKC和MLCK,Ki分别为0.33 μM,1.6 μM,1.6 μM,3.3 μM和36 μM。
Fasudil 103745-39-7 Fasudil hydrochloride (INN) is a potent Rho-kinase inhibitor and vasodilator.
Y-27632 2HCl is a selective ROCK1 (p160ROCK) inhibitor with Ki of 140 nM.
SB 203580;152121-47-6是一种p38 MAPK抑制剂,在THP-1细胞中IC50为0.3-0.5μM,对SAPK3(106T)和SAPK4(106T)选择性低10倍,且阻断PKB磷酸化,IC50为3-5μM。