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CHIR-99021 (CT99021) HCl 1797989-42-4 CHIR-99021 monohydrochloride is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM; 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2,
爱必信特色产品线(全部现货):二抗、标签抗体、对照抗体;WB相关:ECL发光液、预染marker、预制胶;IHC相关:二抗试剂盒、组化笔;IP/CoIP试剂盒;细胞因子、信号通路调节剂;血清、BSA、蛋白酶K、CTB、TTX、CEE;凋亡试剂盒、呼吸爆发试剂盒;动植物提取物...
Cyclosporin A 59865-13-3 CyclosporinA是一种免疫抑制剂,与亲环素结合,随后抑制calcineurin,无细胞试验中IC50为7nM,广泛用于预防器guan移植反应中的排斥反应。
CNQX disodium salt 479347-85-8 CNQX disodium salt is a potent and competitive GluR (kainate/quisqualate (non-NMDA) receptor) antagonist.
CNQX 115066-14-3 CNQX (FG9065) 是高效的 AMPA/kainate 受体拮抗剂。
CHIR-99021 trihydrochloride 1782235-14-6 CHIR-99021 trihydrochloride is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM;
Bortezomib 179324-69-7 Bortezomib is a potent 20S proteasome inhibitor with Ki of 0.6 nM.
BIBF 1120 esylate 656247-18-6 BIBF 1120 esylate是一种有效的 VEGFR1/2/3,FGFR1/2/3 和 PDGFRα/β 三重抑制剂,IC50 值分别为 34 nM/13 nM/13 nM,69 nM/37 nM/108 nM 和 59 nM/65 nM。