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Product Category详细介绍
| 品牌 | absin | 供货周期 | 现货 |
|---|
| 概述 | |
|---|---|
| 描述 | CHIR-99021 is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM; > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases. |
| 别名 | CT99021; CHIR99021; CHIR 99021; CT-99021 |
| 活性 | IC50: 10 nM/6.7 nM (GSK-3α/β) |
| 性能 | |
|---|---|
| 保存方法 | store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. |
| 纯度 | 99% |
| 分子量 | 465.34 |
| 化学式 | C22H18Cl2N8 |
| 分子结构式 | ![]() |
| 溶解性 | DMSO: ≥ 5.1 mg/mL |
| CAS号 | 252917-06-9 |
| 外观 | 粉剂 |
| 功能 | CHIR-99021 是一种 GSK-3α/β 抑制剂,IC50 为 10 nM/6.7 nM。 |
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