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Acalisib (GS-9820) 870281-34-8 Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kδ with IC50 value of 12.7 nM
hPGDS-IN-1 1234708-04-3 hPGDS-IN-1 is a hPGDS inhibitor ,with IC50 of 12 nM in the Fluorescence Polarization Assay or the EIA assay.
AS 602801 848344-36-5 AS 602801(Bentamapimod) is a novel, orally active inhibitor of JNK.
A 438079 hydrochloride 899431-18-6 A-438079 hydrochloride is a potent, and selective P2X7 receptor antagonist with pIC50 of 6.9.
Regadenoson 313348-27-5 Regadenoson is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity.
PIK-75 372196-67-3 PIK-75, a DNA-PK and PI3K inhibitor, suppresses DNA-PK(IC50=2 nM), p110α(IC50=5.8 nM) and p110γ(IC50=76 nM).
Fruquintinib 1194506-26-7 Fruquintinib (HMPL-013) is a small molecule vascular endothelial growth factor receptors inhibitor.
CEP37440 1391712-60-9 CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of 2.3 nM (FAK) and 120 nM(ALK cellular IC50 in 75% human plasma).