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AZD1080 612487-72-6 AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor, inhibits human GSK3α and GSK3β with Ki of 6.9 nM and 31 nM, respectively, shows 14-fold selectivity against
AZD2858 486424-20-8 AZD2858 is a selective GSK-3 inhibitor with an IC50 of 68 nM, activating Wnt signaling, increases bone mass in rats.
CHIR-99021 252917-06-9 CHIR-99021 is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM; 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.
AT13148 1056901-62-2 AT13148 is a novel oral multi-AGC kinase inhibitor with potent pharmacodynamic and antitumor activity, which shows a distinct mechanism of action from other AKT inhibitors.
K-115 223645-67-8 K-115 (free base)是一高效选择性ROCK激酶抑制剂，IC50值为31nM。
GSK269962A(GSK269962) 850664-21-0 GSK269962A(GSK269962)是人ROCK1和ROCK2抑制剂，IC50分别为1.6和4 nM，比对其它丝an酸/苏an酸激酶的抑制性强30倍。
AR-13324 hydrochloride 1253952-02-1 AR-13324是ROCK抑制剂，Ki值为0.2-10.3 nM。
Fasudil hydrochloride 105628-07-7 Fasudil Hydrochloride (盐suan法舒地尔; HA-1077; AT-877) 能抑制ROCK-II，PKA，PKG，PKC和MLCK，Ki分别为0.33 μM，1.6 μM，1.6 μM，3.3 μM和36 μM。
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